Micro-photo-flow reactor system for fused N-heteroaryl scaffold synthesis and late-stage functionalization of pyrazolopyridines-Reference-Cited by-同舟云学术

Micro-photo-flow reactor system for fused N-heteroaryl scaffold synthesis and late-stage functionalization of pyrazolopyridines

Published:2022 Issue:80 Volume:58 Page:11268-11271
ISSN:1359-7345
Container-title:Chemical Communications
language:en
Short-container-title:Chem. Commun.

Author:

Kumar Sanjeev¹²,Singh Ajay K.¹²^ORCID

Affiliation:

1. Department of Organic Synthesis and Process Chemistry, CSIR-Indian Institute of Chemical Technology, Hyderabad-500007, India

2. Academy of Scientific and Innovative Research (AcSIR), Ghaziabad 201002, Uttar Pradesh, India

Abstract

Late-stage functionalization (LSF) of active pharmaceutical ingredients can provide a straightforward approach to efficient de novo design and synthesis of drug molecules for structural activity relationship studies (SARS).

Funder

Council of Scientific and Industrial Research, India

Publisher

Royal Society of Chemistry (RSC)

Subject

Materials Chemistry,Metals and Alloys,Surfaces, Coatings and Films,General Chemistry,Ceramics and Composites,Electronic, Optical and Magnetic Materials,Catalysis

Link

http://pubs.rsc.org/en/content/articlepdf/2022/CC/D2CC03713K

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3. Asymmetric Intramolecular Dearomatization of Nonactivated Arenes with Ynamides for Rapid Assembly of Fused Ring System under Silver Catalysis

4. Palladium-Catalyzed [3 + 2] Annulation of Alkynes with Concomitant Aromatic Ring Expansion: A Concise Approach to (Pseudo)azulenes

5. Photoinduced ynamide structural reshuffling and functionalization

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