Transition metal-free aminofluorination of β,γ-unsaturated hydrazones: base-controlled regioselective synthesis of fluorinated dihydropyrazole and tetrahydropyridazine derivatives
Author:
Affiliation:
1. Key Laboratory of Organofluorine Chemistry
2. Shanghai Institute of Organic Chemistry
3. University of Chinese Academy of Sciences
4. Chinese Academy of Sciences
5. Shanghai 200032
Abstract
Various base-controlled regioselective reactions of β,γ-unsaturated hydrazones with Selectfluor were achieved under transition metal-free conditions.
Funder
National Natural Science Foundation of China
Science and Technology Commission of Shanghai Municipality
Publisher
Royal Society of Chemistry (RSC)
Subject
Organic Chemistry
Link
http://pubs.rsc.org/en/content/articlepdf/2018/QO/C7QO01105A
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4. Fluorine in Pharmaceuticals: Looking Beyond Intuition
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