Pyrazolobenzothiazine-based carbothioamides as new structural leads for the inhibition of monoamine oxidases: design, synthesis, in vitro bioevaluation and molecular docking studies-Reference-Cited by-同舟云学术

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Pyrazolobenzothiazine-based carbothioamides as new structural leads for the inhibition of monoamine oxidases: design, synthesis, in vitro bioevaluation and molecular docking studies

Published:2017 Issue:2 Volume:8 Page:452-464
ISSN:2040-2503
Container-title:MedChemComm
language:en
Short-container-title:Med. Chem. Commun.

Author:

Abid Syed Mobasher Ali¹²³⁴,Aslam Sana⁵⁶⁷⁴⁸,Zaib Sumera¹²³⁴,Bakht Syeda Mahwish¹²³⁴,Ahmad Matloob⁵⁹⁷⁴,Athar Muhammad Makshoof⁸¹⁰¹¹⁴,Gardiner John M.¹²¹³¹⁴¹⁵,Iqbal Jamshed¹²³⁴^ORCID

Affiliation:

1. Centre for Advanced Drug Research

2. COMSATS Institute of Information Technology

3. Abbottabad-22060

4. Pakistan

5. Department of Chemistry

6. Government College Women University

7. Faisalabad-38000

8. Institute of Chemistry

9. Government College University

10. University of the Punjab

11. Lahore

12. School of Chemistry and Manchester Institute of Biotechnology

13. University of Manchester

14. Manchester M1 7DN

15. UK

Abstract

Binding mode of potent inhibitor (green) & cognate ligand (pink) in the active site of MAO-B.

Funder

Higher Education Commission, Pakistan

Publisher

Royal Society of Chemistry (RSC)

Subject

Pharmaceutical Science,Biochemistry,Drug Discovery,Molecular Medicine,Pharmacology,Organic Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2017/MD/C6MD00570E

Reference31 articles.

1. Discovery of New Chemical Entities for Old Targets: Insights on the Lead Optimization of Chromone-Based Monoamine Oxidase B (MAO-B) Inhibitors

2. Monoamine Oxidase Inhibition and Molecular Modeling Studies of Piperidyl-thienyl and 2-Pyrazoline Derivatives of Chalcones

3. Proposed interaction of some novel antidepressant pyrazolines against monoamine oxidase isoforms. Molecular docking studies and PASS assisted in silico approach

4. Localization of distinct monoamine oxidase a and monoamine oxidase b cell populations in human brainstem

5. Interactions of Nitrogen-Containing Xenobiotics with Monoamine Oxidase (MAO) Isozymes A and B: SAR Studies on MAO Substrates and Inhibitors

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4. Perchlorate-induced structural diversity in thiosemicarbazone copper(ii) complexes provides insights to understand the reactivity in acidic and basic media;CrystEngComm;2023

5. Recent Advances in Synthesis and Medicinal Evaluation of 1,2‐Benzothiazine Analogues;Asian Journal of Organic Chemistry;2022-06-24

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