Borylated cyclobutanes <i>via</i> thermal [2 + 2]-cycloaddition-Reference-Cited by-同舟云学术

Borylated cyclobutanes via thermal [2 + 2]-cycloaddition

Published:2024 Issue:9 Volume:15 Page:3249-3254
ISSN:2041-6520
Container-title:Chemical Science
language:en
Short-container-title:Chem. Sci.

Author:

Prysiazhniuk Kateryna¹,Polishchuk Oleksandr¹,Shulha Stanislav¹,Gudzikevych Kyrylo¹,Datsenko Oleksandr P.¹,Kubyshkin Vladimir¹^ORCID,Mykhailiuk Pavel K.¹^ORCID

Affiliation:

1. Enamine Ltd, Winston Churchill St. 78, 02094 Kyiv, Ukraine

Abstract

A one-step approach to borylated cyclobutanes from amides of carboxylic acids and vinyl boronates is elaborated. The reaction proceeds via the thermal [2 + 2]-cycloaddition of in situ-generated keteniminium salts.

Funder

H2020 European Research Council

Publisher

Royal Society of Chemistry (RSC)

Link

http://pubs.rsc.org/en/content/articlepdf/2024/SC/D3SC06600B

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