Quantification of crystallinity during indomethacin crystalline transformation from α- to γ-polymorphic forms and of the thermodynamic contribution to dissolution in aqueous buffer and solutions of solubilizer-Reference-Cited by-同舟云学术

Quantification of crystallinity during indomethacin crystalline transformation from α- to γ-polymorphic forms and of the thermodynamic contribution to dissolution in aqueous buffer and solutions of solubilizer

Published:2024 Issue:6 Volume:14 Page:4129-4141
ISSN:2046-2069
Container-title:RSC Advances
language:en
Short-container-title:RSC Adv.

Author:

Hasegawa Kanji¹,Goto Satoru¹^ORCID,Kataoka Hikaru¹^ORCID,Chatani Hitoshi¹,Kinoshita Takatoshi¹,Yokoyama Hideshi¹,Tsuchida Tomohiro¹^ORCID

Affiliation:

1. Faculty of Pharmaceutical Sciences, Tokyo University of Science, 2641 Yamazaki, Noda, Chiba 278-8510, Japan

Abstract

The thermodynamic properties and dissolution of indomethacin (INM) were analyzed as models for poorly water-soluble drugs.

Publisher

Royal Society of Chemistry (RSC)

Link

http://pubs.rsc.org/en/content/articlepdf/2024/RA/D3RA08481G

Reference63 articles.

1. Regulatory considerations of pharmaceutical solid polymorphism in Abbreviated New Drug Applications (ANDAs)

2. Physical and chemical stability of drug nanoparticles

3. Unlocking the potential of drug-drug cocrystals – A comprehensive review

4. Dry mechanochemical synthesis of ethenzamide and saccharin 1:1 cocrystal and their evaluation using powder X-ray diffraction and FT-MIR and NIR spectroscopy

5. Polymeric Amorphous Solid Dispersions: A Review of Amorphization, Crystallization, Stabilization, Solid-State Characterization, and Aqueous Solubilization of Biopharmaceutical Classification System Class II Drugs

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