Photoredox Ni-catalyzed peptide C(sp2)–O cross-coupling: from intermolecular reactions to side chain-to-tail macrocyclization
Author:
Affiliation:
1. Department of Discovery Chemistry
2. MRL
3. Merck & Co., Inc.
4. Boston
5. USA
6. Computational and Structural Chemistry
7. Kenilworth
8. Process and Analytical Research and Development
9. Chemistry Capabilities for Accelerating Therapeutics
Abstract
Ni/photoredox (4DPAIPN) dual catalysis enabled challenging peptide C(sp2)–O coupling reactions.
Funder
Merck
Publisher
Royal Society of Chemistry (RSC)
Subject
General Chemistry
Link
http://pubs.rsc.org/en/content/articlepdf/2019/SC/C9SC00694J
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