Synthesis, biological and molecular modelling for 1,3,4-thiadiazole sulfonyl thioureas: bacterial and fungal activity-Reference-Cited by-同舟云学术

Synthesis, biological and molecular modelling for 1,3,4-thiadiazole sulfonyl thioureas: bacterial and fungal activity

Published:2023 Issue:12 Volume:14 Page:2751-2767
ISSN:2632-8682
Container-title:RSC Medicinal Chemistry
language:en
Short-container-title:RSC Med. Chem.

Author:

Dinh Thanh Nguyen¹^ORCID,Ngoc Toan Vu¹²,Thi Kim Giang Nguyen¹³,Thi Kim Van Hoang¹⁴,Son Hai Do¹³,Minh Tri Nguyen¹³,Ngoc Toan Duong¹⁵

Affiliation:

1. Faculty of Chemistry, University of Science (Vietnam National University, Hanoi), 19 Le Thanh Tong, Ha Noi, Viet Nam

2. Institute of New Technology, Military Institute of Science and Technology (Ministry of Military), 17 Hoang Sam, Cau Giay, Ha Noi, Viet Nam

3. Institute of Science and Technology, Ministry of Public Security of Vietnam, 47 Pham Van Dong, Cau Giay, Ha Noi, Vietnam

4. Faculty of Chemical Technology, Viet Tri University of Industry, Tien Kien, Lam Thao, Phu Tho, Viet Nam

5. Faculty of Chemistry, Thai Nguyen University of Education, 20 Luong Ngoc Quyen, Thai Nguyen, Viet Nam

Abstract

Sulfonylthioureas of 2-amino-1,3-thiadiazoles and 4-toluenesulfonyl isocyanate had inhibitions for bacteria, fungi, S. aureus DNA gyrase, TopoIV and DHF reductase. IFD, MM-GBSA and MD were performed.

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Drug Discovery,Pharmaceutical Science,Pharmacology,Molecular Medicine,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2023/MD/D3MD00508A

Reference55 articles.

1. S.Doron and S. L.Gorbach , in International Encyclopedia of Public Health , ed. H. K. Heggenhougen , Academic Press, Oxford , 2008 , pp. 273–282 , 10.1016/B978-012373960-5.00596-7

2. 1,3,4-Thiadiazole: Synthesis, Reactions, and Applications in Medicinal, Agricultural, and Materials Chemistry

3. 1,3,4-Thiadiazole and its Derivatives: A Review on Recent Progress in Biological Activities

4. Diverse Biological Activities of 1,3,4-Thiadiazole Scaffold

5. Thiadiazole derivatives as anticancer agents

Cited by 1 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Synthesis and biological evaluation of new naphthalimide–thiourea derivatives as potent antimicrobial agents active against multidrug-resistant Staphylococcus aureus and Mycobacterium tuberculosis;RSC Medicinal Chemistry;2024