Novel 1,2,4-oxadiazole compounds as PPAR-α ligand agonists: a new strategy for the design of antitumour compounds

Author:

Apaza Ticona Luis12ORCID,Sánchez Sánchez-Corral Javier2,Flores Sepúlveda Alejandro3ORCID,Soriano Vázquez Carmen3,Hernán Vieco Carmen3ORCID,Rumbero Sánchez Ángel2

Affiliation:

1. Organic Chemistry Unit, Department of Chemistry in Pharmaceutical Sciences, Faculty of Pharmacy, Universidad Complutense of Madrid, Plaza Ramón y Cajal s/n, 28040 Madrid, Spain

2. Department of Organic Chemistry, Faculty of Sciences, University Autónoma of Madrid, Cantoblanco, 28040 Madrid, Spain

3. Faculty of Pharmacy, Universidad Complutense of Madrid, Plaza Ramón y Cajal s/n, 28040 Madrid, Spain

Abstract

Modulation of PPAR-α by natural ligands is a novel strategy for the development of anticancer therapies.

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Drug Discovery,Pharmaceutical Science,Pharmacology,Molecular Medicine,Biochemistry

Reference44 articles.

1. Cancer , https://www.who.int/es/news-room/fact-sheets/detail/cancer , (accessed 3 December 2022 )

2. Effects of acupuncture on cancer-related fatigue: a meta-analysis

3. Cancer statistics, 2020

4. The Role of PPARs in Disease

5. The Role of PPARs in Cancer

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