Stereoselective synthesis of all-cis boryl tetrahydroquinolines via copper-catalyzed regioselective addition/cyclization of o-aldiminyl cinnamate with B2Pin2-Reference-Cited by-同舟云学术

Stereoselective synthesis of all-cis boryl tetrahydroquinolines via copper-catalyzed regioselective addition/cyclization of o-aldiminyl cinnamate with B2Pin2

Published:2019 Issue:6 Volume:17 Page:1542-1546
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Bi Ya-Ping¹²³⁴⁵,Wang He-Min¹²³⁴⁵,Qu Hong-Yu¹²³⁴⁵,Liang Xian-Chen¹²³⁴⁵,Zhou Ying¹²³⁴⁵,Li Xue-Ying¹²³⁴⁵,Xu Defeng¹²³⁴⁵,Shen Mei-Hua¹²³⁴⁵^ORCID,Xu Hua-Dong¹²³⁴⁵^ORCID

Affiliation:

1. Jiangsu Key Laboratory of Advanced Catalytic Materials & Technology

2. School of Pharmaceutical Engineering and Life Science

3. Changzhou University

4. Changzhou

5. China

Abstract

All-cis 2-aryl-3-carboxylate-4-boryl tetrahydroquinolines can be made exclusively via a copper-catalyzed carboboration of aryl acrylates with aldimines.

Funder

National Natural Science Foundation of China

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2019/OB/C8OB03195A

Reference62 articles.

1. Recent Advances in the DABOs Family as Potent HIV-1 non-Nucleoside Reverse Transcriptase Inhibitors

2. Recent progress in the synthesis of 1,2,3,4,-tetrahydroquinolines

3. Protective Effect of Qnr on Agents Other than Quinolones That Target DNA Gyrase