Synthesis, characterization and biological activity of fluorescently labeled bedaquiline analogues-Reference-Cited by-同舟云学术

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Synthesis, characterization and biological activity of fluorescently labeled bedaquiline analogues

Published:2016 Issue:110 Volume:6 Page:108708-108716
ISSN:2046-2069
Container-title:RSC Advances
language:en
Short-container-title:RSC Adv.

Author:

Rombouts Jeroen A.¹²³⁴⁵,Veenboer Richard M. P.¹²³⁴,Villellas Cristina⁶⁷⁸⁹¹⁰,Lu Ping¹¹¹²¹³²³,Ehlers Andreas W.¹²³⁴¹⁴,Andries Koen⁶⁷⁸⁹¹⁰,Koul Anil⁶⁷⁸⁹¹⁰,Lill Holger¹¹¹²¹³²³,Ruijter Eelco⁵¹⁵²¹⁶⁴^ORCID,Orru Romano V. A.⁵¹⁵²¹⁶⁴,Lammertsma Koop¹²³⁴¹⁴,Bald Dirk¹¹¹²¹³²³,Slootweg J. Chris¹²³⁴

Affiliation:

1. Department of Chemistry and Pharmaceutical Sciences

2. Vrije Universiteit Amsterdam

3. 1081 HV Amsterdam

4. The Netherlands

5. Department of Chemistry & Pharmaceutical Sciences

6. Infectious Diseases and Vaccines Therapeutic Area

7. Janssen Research & Development

8. Johnson & Johnson Pharmaceuticals

9. 2340 Beerse

10. Belgium

11. Department of Molecular Cell Biology

12. AIMMS

13. Faculty of Earth and Life Sciences

14. Department of Chemistry

15. Amsterdam Institute for Molecules Medicines and Systems (AIMMS)

16. 1081 HZ Amsterdam

Abstract

Labeling the tuberculosis drug bedaquiline with a fluorescent alkynyl-BODIPY moiety does not disrupt its antibacterial properties.

Funder

VU University Amsterdam

Publisher

Royal Society of Chemistry (RSC)

Subject

General Chemical Engineering,General Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2016/RA/C6RA22693K

Reference41 articles.

1. World Health Organization , Global tuberculosis report 2015, World Health Organization, 2015

2. The challenge of new drug discovery for tuberculosis

3. Respiratory ATP synthesis: the new generation of mycobacterial drug targets?

4. Targeting bacterial membrane function: an underexploited mechanism for treating persistent infections

5. Energy Metabolism and Drug Efflux in Mycobacterium tuberculosis

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2. Synthesis, Characterization, and Stability Assessment for the Benzoate, Hydrochloride, Malonate, and Nicotinate Salts of Bedaquiline;Pharmaceuticals;2023-02-08

3. Quinoline Hydrazide/Hydrazone Derivatives: Recent Insights on Antibacterial Activity and Mechanism of Action;ChemMedChem;2023-01-20

4. Salts and Polymorph Screens for Bedaquiline;AAPS PharmSciTech;2021-08-25

5. Evaluation of physicochemical stability and degradation kinetics of bedaquiline in hydrolytic solutions of different pH;Future Journal of Pharmaceutical Sciences;2021-04-14

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