Domino reaction of cyclic sulfamidate imines with Morita–Baylis–Hillman acetates promoted by DABCO: a metal-free approach to functionalized nicotinic acid derivatives

Author:

Majee Debashis1234,Biswas Soumen1234,Mobin Shaikh M.1234ORCID,Samanta Sampak1234ORCID

Affiliation:

1. Discipline of Chemistry

2. Indian Institute of Technology Indore

3. Simrol

4. India

Abstract

A series of 4,6-diarylnicotinates have been prepared in good to excellent yields via a domino reaction of cyclic sulfamidate imines with MBH acetates in 2-MeTHF promoted by DABCO under an O2 atmosphere.

Funder

Science and Engineering Research Board

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Reference56 articles.

1. H. L. Fraser , D. W.Hopper, K. M. K.Kutterer and A. L.Crombie, in Progress in Heterocyclic Chemistry, ed. G. W. Gribble and J. A. Joule, Elsevier, Amsterdam, 2008, vol. 19, p. 314

2. An overview of the synthetic routes to the best selling drugs containing 6-membered heterocycles

3. Metal-Free Multicomponent Syntheses of Pyridines

4. Recent Strategies for the Synthesis of Pyridine Derivatives

5. Investigating the continuous synthesis of a nicotinonitrile precursor to nevirapine

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