Synthesis and amylin receptor activity of glycomimetics of pramlintide using click chemistry-Reference-Cited by-同舟云学术

Synthesis and amylin receptor activity of glycomimetics of pramlintide using click chemistry

Published:2016 Issue:23 Volume:14 Page:5238-5245
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Yule Lauren R.¹²³⁴⁵,Bower Rebekah L.¹²³⁴,Kaur Harveen⁵²³⁴⁶,Kowalczyk Renata¹²³⁴⁵,Hay Debbie L.¹²³⁴⁶,Brimble Margaret. A.¹²³⁴⁵

Affiliation:

1. The School of Biological Sciences

2. University of Auckland

3. Auckland 1010

4. New Zealand

5. The School of Chemical Sciences

6. Maurice Wilkins Centre for Molecular Biodiscovery

Abstract

Synthetic clicked pramlintide glycomimetics maintained AMY_1(a)activity and are expected to possess superior synthetic and pharmacokinetic properties thanN-glycosylated analogues.

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2016/OB/C6OB00850J

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4. Long-Acting Glucagon-Like Peptide 1 Receptor Agonists

5. Activity of Pramlintide, Rat and Human Amylin but not Aβ1–42 at Human Amylin Receptors

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