Advances in the development of pyridinone derivatives as non-nucleoside reverse transcriptase inhibitors-Reference-Cited by-同舟云学术

Advances in the development of pyridinone derivatives as non-nucleoside reverse transcriptase inhibitors

Published:2016 Issue:3 Volume:6 Page:2119-2130
ISSN:2046-2069
Container-title:RSC Advances
language:en
Short-container-title:RSC Adv.

Author:

Vite-Caritino Hugo¹²³⁴⁵,Méndez-Lucio Oscar⁶⁷⁸⁹¹⁰,Reyes Héctor¹¹¹²⁵,Cabrera Alberto¹¹¹²⁵,Chávez Daniel¹¹¹²⁵,Medina-Franco José L.¹²³⁴⁵^ORCID

Affiliation:

1. Facultad de Química

2. Departamento de Farmacia

3. Universidad Nacional Autónoma de México

4. Mexico City 04510

5. Mexico

6. Unilever Centre for Molecular Science Informatics

7. Department of Chemistry

8. University of Cambridge

9. Cambridge CB2 1EW

10. UK

11. Centro de Graduados e Investigación en Química del Instituto Tecnológico de Tijuana

12. Tijuana

Abstract

Medicinal chemistry, computational design and biological screening have advanced pyridin-2(1H)-one derivatives as a promising class of non-nucleoside reverse transcriptase inhibitors for the treatment of HIV/AIDS.

Funder

Consejo Nacional de Ciencia y Tecnología

Publisher

Royal Society of Chemistry (RSC)

Subject

General Chemical Engineering,General Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2016/RA/C5RA25722K

Reference43 articles.

1. World Health Organization , HIV/AIDS, availale at http://www.who.int/hiv/data/en/

2. Non-nucleoside reverse transcriptase inhibitors (NNRTIs), their discovery, development, and use in the treatment of HIV-1 infection: A review of the last 20 years (1989–2009)

3. The Protein Data Bank

4. Crystal Structure at 3.5 Å Resolution of HIV-1 Reverse Transcriptase Complexed with an Inhibitor

5. NMR characterization of HIV-1 reverse transcriptase binding to various non-nucleoside reverse transcriptase inhibitors with different activities

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