Selective access to dipyrazolo-fused pyridines via formal [3 + 2 + 1] heteroannulation of methyl ketones with pyrazol-5-amines
Author:
Affiliation:
1. School of Pharmacy
2. Xinxiang Medical University
3. Xinxiang
4. P. R. China
5. Key Laboratory of Pesticide & Chemical Biology
6. Ministry of Education
7. College of Chemistry
8. Central China Normal University
9. Wuhan 430079
Abstract
A fascinating new form of the Hantzsch reaction with methyl ketones and pyrazol-5-amines for the selective synthesis of dipyrazolo-fused pyridines has been discovered.
Publisher
Royal Society of Chemistry (RSC)
Subject
Organic Chemistry
Link
http://pubs.rsc.org/en/content/articlepdf/2018/QO/C7QO00941K
Reference36 articles.
1. Interferon inducing activities of derivatives of 1,3-dimethyl-4-(3-dimethylaminopropylamino)-1H-pyrazolo[3,4-b]quinoline and related compounds
2. Pyrazoloheteroaryls: Novel p38α MAP kinase inhibiting scaffolds with oral activity
3. Substituted Pyrazolo[3,4-b]pyridines as Potent A1 Adenosine Antagonists: Synthesis, Biological Evaluation, and Development of an A1 Bovine Receptor Model
4. Antimalarials. 4-Substituted 1H-pyrazolo[3,4-b]quinolines
5. Pyrazolopyridine inhibitors of B-RafV600E. Part 2: Structure–activity relationships
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