Transition metal-free direct trifluoromethylthiolation of indoles using trifluoromethanesulfonyl chloride in the presence of triphenylphosphine-Reference-Cited by-同舟云学术

Transition metal-free direct trifluoromethylthiolation of indoles using trifluoromethanesulfonyl chloride in the presence of triphenylphosphine

Published:2017 Issue:5 Volume:15 Page:1254-1260
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Lu Kui¹²³⁴⁵^ORCID,Deng Zhijie⁶⁷⁸⁹¹⁰,Li Ming¹²³⁴⁵,Li Tianjiao⁶⁷⁸⁹¹⁰,Zhao Xia⁶⁷⁸⁹¹⁰

Affiliation:

1. China International Science and Technology Cooperation Base of Food Nutrition/Safety and Medicinal Chemistry

2. Key Laboratory of Industrial Microbiology of Ministry of Education

3. Tianjin Key Laboratory of Industry Microbiology

4. College of Biotechnology

5. Tianjin University of Science & Technology

6. College of Chemistry

7. Tianjin Key Laboratory of Structure and Performance for Functional Molecules

8. Key laboratory of Inorganic–Organic Hybrid Functional Material Chemistry

9. Ministry of Education

10. Tianjin Normal University

Abstract

A novel triphenylphosphine-mediated direct trifluoromethylthiolation of indole derivatives using trifluoromethanesulfonyl chloride as the SCF₃ source was developed.

Funder

National Natural Science Foundation of China

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2017/OB/C6OB02465C

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