Synthesis of bridgehead-azacycles <i>via</i> dual C–N/C–C annulation of α-amino acids, aminals and maleimides-Reference-Cited by-同舟云学术

Synthesis of bridgehead-azacycles via dual C–N/C–C annulation of α-amino acids, aminals and maleimides

Published:2022 Issue:32 Volume:20 Page:6368-6383
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Thadem Nagender¹²,Rajesh Manda¹^ORCID,Balaboina Harikrishna¹,Das Saibal¹²^ORCID

Affiliation:

1. Department of Organic Synthesis & Process Chemistry, CSIR-Indian Institute of Chemical Technology (CSIR-IICT), Hyderabad 500007, India

2. Academy of Scientific and Innovative Research (AcSIR), Ghaziabad, 201002, India

Abstract

A rare dipolarophile-induced diastereo-selective amidative annulation and concomitant 3 + 2 cycloaddition are reported using α-amino acids, amino aldehydes and maleimides.

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2022/OB/D2OB01117D

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