Structural basis for modulation of a G-protein-coupled receptor by allosteric drugs-Reference-Cited by-同舟云学术

Structural basis for modulation of a G-protein-coupled receptor by allosteric drugs

Published:2013-10-13 Issue:7475 Volume:503 Page:295-299
ISSN:0028-0836
Container-title:Nature
language:en
Short-container-title:Nature

Author:

Dror Ron O.,Green Hillary F.,Valant Celine,Borhani David W.,Valcourt James R.,Pan Albert C.,Arlow Daniel H.,Canals Meritxell,Lane J. Robert,Rahmani Raphaël,Baell Jonathan B.,Sexton Patrick M.,Christopoulos Arthur,Shaw David E.

Publisher

Springer Science and Business Media LLC

Subject

Multidisciplinary

Link

http://www.nature.com/articles/nature12595.pdf

Reference53 articles.

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2. Keov, P., Sexton, P. M. & Christopoulos, A. Allosteric modulation of G protein-coupled receptors: a pharmacological perspective. Neuropharmacology 60, 24–35 (2011)

3. Filmore, D. It’s a GPCR world. Modern Drug Discov. 7, 24–28 (2004)

4. Jakubik, J. & El-Fakahany, E. E. Allosteric modulation of muscarinic acetylcholine receptors. Pharmaceuticals 3, 2838–2860 (2010)

5. Haga, K. et al. Structure of human M2 muscarinic acetylcholine receptor bound to an antagonist. Nature 482, 547–551 (2012)

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