Discovery of novel antagonists targeting the DNA binding domain of androgen receptor by integrated docking-based virtual screening and bioassays-Reference-Cited by-同舟云学术

Discovery of novel antagonists targeting the DNA binding domain of androgen receptor by integrated docking-based virtual screening and bioassays

Published:2021-03-25 Issue:1 Volume:43 Page:229-239
ISSN:1671-4083
Container-title:Acta Pharmacologica Sinica
language:en
Short-container-title:Acta Pharmacol Sin

Author:

Pang Jin-ping,Shen Chao,Zhou Wen-fang,Wang Yun-xia,Shan Lu-hu,Chai Xin,Shao Ying,Hu Xue-ping,Zhu Feng,Zhu Dan-yan,Xiao Li,Xu Lei,Xu Xiao-hong,Li Dan,Hou Ting-jun

Publisher

Springer Science and Business Media LLC

Subject

Pharmacology (medical),Pharmacology,General Medicine

Link

https://www.nature.com/articles/s41401-021-00632-5.pdf

Reference60 articles.

1. Huggins C, Stevens RE, Hodges CV. Studies on prostate cancer II the effects of castration on advanced carcinoma of the prostate gland. Arch Surg-Chic. 1941;43:209–23.

2. Bohl CE, Gao WQ, Miller DD, Bell CE, Dalton JT. Structural basis for antagonism and resistance of bicalutamide in prostate cancer. Proc Natl Acad Sci USA. 2005;102:6201–6.

3. Li YM, Chan SC, Brand LJ, Hwang TH, Silverstein KAT, Dehm SM. Androgen receptor splice variants mediate enzalutamide resistance in castration-resistant prostate cancer cell lines. Cancer Res. 2013;73:483–9.

4. Li D, Zhou WF, Pang JP, Tang Q, Zhong BL, Shen C, et al. A magic drug target: androgen receptor. Med Res Rev. 2019;39:1485–514.

5. Chen CD, Welsbie DS, Tran C, Baek SH, Chen R, Vessella R, et al. Molecular determinants of resistance to antiandrogen therapy. Nat Med. 2004;10:33–9.

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