Structural basis of GABA reuptake inhibition-Reference-Cited by-同舟云学术

Structural basis of GABA reuptake inhibition

Published:2022-06-08 Issue:7915 Volume:606 Page:820-826
ISSN:0028-0836
Container-title:Nature
language:en
Short-container-title:Nature

Author:

Motiwala Zenia^ORCID,Aduri Nanda Gowtham,Shaye Hamidreza,Han Gye Won,Lam Jordy Homing,Katritch Vsevolod^ORCID,Cherezov Vadim^ORCID,Gati Cornelius^ORCID

Publisher

Springer Science and Business Media LLC

Subject

Multidisciplinary

Link

https://www.nature.com/articles/s41586-022-04814-x.pdf

Reference72 articles.

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3. Braestrup, C. et al. (R)-N-[4,4-bis(3-methyl-2-thienyl)but-3-en-1-yl]nipecotic acid binds with high affinity to the brain gamma-aminobutyric acid uptake carrier. J. Neurochem. 54, 639–647 (1990).

4. Blat, Y. Non-competitive inhibition by active site binders. Chem. Biol. Drug Des. 75, 535–540 (2010).

5. Sieghart, W. Structure, pharmacology, and function of GABAA receptor rubtypes. GABA 54, 231–263 (2006).

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