A three-stage biophysical screening cascade for fragment-based drug discovery-Reference-Cited by-同舟云学术

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A three-stage biophysical screening cascade for fragment-based drug discovery

Published:2013-10-24 Issue:11 Volume:8 Page:2309-2324
ISSN:1754-2189
Container-title:Nature Protocols
language:en
Short-container-title:Nat Protoc

Author:

Mashalidis Ellene H,Śledź Paweł,Lang Steffen,Abell Chris

Publisher

Springer Science and Business Media LLC

Subject

General Biochemistry, Genetics and Molecular Biology

Link

http://www.nature.com/articles/nprot.2013.130.pdf

Reference62 articles.

1. Murray, C.W. & Rees, D.C. The rise of fragment-based drug discovery. Nat. Chem. 1, 187–192 (2009).

2. Ciulli, A. & Abell, C. Fragment-based approaches to enzyme inhibition. Curr. Opin. Biotechnol. 18, 489–496 (2007).

3. Congreve, M., Carr, R., Murray, C. & Jhoti, H. A 'rule of three' for fragment-based lead discovery? Drug Discov. Today 8, 876–877 (2003).

4. Hung, A. et al. Application of fragment growing and fragment linking to the discovery of inhibitors of Mycobacterium tuberculosis pantothenate synthetase. Angew. Chem. Int. Ed. 48, 8452–8456 (2009).

5. Hudson, S.A. et al. Application of fragment screening and merging to the discovery of inhibitors of the Mycobacterium tuberculosis cytochrome P450 CYP121. Angew. Chem. Int. Ed. 51, 9311–9316 (2012).

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