Targeting ErbB2 and ErbB3 with a bispecific single-chain Fv enhances targeting selectivity and induces a therapeutic effect in vitro

Author:

Robinson M K,Hodge K M,Horak E,Sundberg Å L,Russeva M,Shaller C C,von Mehren M,Shchaveleva I,Simmons H H,Marks J D,Adams G P

Publisher

Springer Science and Business Media LLC

Subject

Cancer Research,Oncology

Reference63 articles.

1. Adams GP, McCartney JE, Tai M-S, Oppermann H, Huston JS, Stafford WF, Bookman MA, Fand I, Houston LL, Weiner LM (1993) Highly specific in vivo tumor targeting by monovalent and divalent forms of 741F8 anti-c-erbB-2 single-chain Fv. Cancer Res 53: 4026–4034

2. Adams GP, Schier R, Marshall K, Wolf EJ, McCall AM, Marks JD, Weiner LM (1998) Increased affinity leads to improved selective tumor delivery of single-chain Fv antibodies. Cancer Res 58: 485–490

3. Adams GP, Tai MS, McCartney JE, Marks JD, Stafford III WF, Houston LL, Huston JS, Weiner LM (2006) Avidity-mediated enhancement of in vivo tumor targeting by single-chain Fv dimers. Clin Cancer Res 12 (5): 1599–1605

4. Adams GP, Weiner LM (2005) Monoclonal antibody therapy of cancer. Nat Biotechnol 23 (9): 1147–1157

5. Agus DB, Akita RW, Fox WD, Lewis GD, Higgins B, Pisacane PI, Lofgren JA, Tindell C, Evans DP, Maiese K (2002) Targeting ligand-activated ErbB2 signaling inhibits breast and prostate tumor growth. Cancer Cell 2 (2): 127–137

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