Conformational Selection and Induced Fit Mechanisms in the Binding of an Anticancer Drug to the c-Src Kinase-Reference-Cited by-同舟云学术

Conformational Selection and Induced Fit Mechanisms in the Binding of an Anticancer Drug to the c-Src Kinase

Published:2016-04 Issue:1 Volume:6 Page:
ISSN:2045-2322
Container-title:Scientific Reports
language:en
Short-container-title:Sci Rep

Author:

Morando Maria Agnese,Saladino Giorgio,D’Amelio Nicola,Pucheta-Martinez Encarna,Lovera Silvia,Lelli Moreno,López-Méndez Blanca,Marenchino Marco,Campos-Olivas Ramón,Gervasio Francesco Luigi

Publisher

Springer Science and Business Media LLC

Subject

Multidisciplinary

Link

http://www.nature.com/articles/srep24439.pdf

Reference57 articles.

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4. Hammes, G. G., Chang, Y.-C. & Oas, T. G. Conformational selection or induced fit: a flux description of reaction mechanism. Proc. Natl. Acad. Sci. USA 106, 13737–13741 (2009).

5. D’Abramo, M., Rabal, O., Oyarzabal, J. & Gervasio, F. L. Conformational Selection versus Induced Fit in Kinases: The Case of PI3K-γ. Angew. Chem. Int. Ed. 124, 666–670 (2012).

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