Structural basis of small-molecule inhibition of human multidrug transporter ABCG2-Reference-Cited by-同舟云学术

Structural basis of small-molecule inhibition of human multidrug transporter ABCG2

Published:2018-04 Issue:4 Volume:25 Page:333-340
ISSN:1545-9993
Container-title:Nature Structural & Molecular Biology
language:en
Short-container-title:Nat Struct Mol Biol

Author:

Jackson Scott M.^ORCID,Manolaridis Ioannis,Kowal Julia^ORCID,Zechner Melanie,Taylor Nicholas M. I.^ORCID,Bause Manuel,Bauer Stefanie,Bartholomaeus Ruben,Bernhardt Guenther,Koenig Burkhard,Buschauer Armin,Stahlberg Henning^ORCID,Altmann Karl-Heinz,Locher Kaspar P.^ORCID

Publisher

Springer Science and Business Media LLC

Subject

Molecular Biology,Structural Biology

Link

http://www.nature.com/articles/s41594-018-0049-1.pdf

Reference67 articles.

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3. Fetsch, P. A. et al. Localization of the ABCG2 mitoxantrone resistance-associated protein in normal tissues. Cancer Lett. 235, 84–92 (2006).

4. Robey, R. W. et al. ABCG2: a perspective. Adv. Drug Deliv. Rev. 61, 3–13 (2009).

5. Ishikawa, T., Aw, W. & Kaneko, K. Metabolic interactions of purine derivatives with human ABC transporter ABCG2: genetic testing to assess gout risk. Pharmaceuticals (Basel) 6, 1347–1360 (2013).

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