Inactive and active state structures template selective tools for the human 5-HT5A receptor-Reference-Cited by-同舟云学术

Inactive and active state structures template selective tools for the human 5-HT5A receptor

Published:2022-07 Issue:7 Volume:29 Page:677-687
ISSN:1545-9993
Container-title:Nature Structural & Molecular Biology
language:en
Short-container-title:Nat Struct Mol Biol

Author:

Zhang Shicheng^ORCID,Chen He,Zhang Chengwei,Yang Ying,Popov Petr,Liu Jing^ORCID,Krumm Brian E.^ORCID,Cao Can^ORCID,Kim Kuglae,Xiong Yan,Katritch Vsevolod^ORCID,Shoichet Brian K.^ORCID,Jin Jian^ORCID,Fay Jonathan F.^ORCID,Roth Bryan L.^ORCID

Publisher

Springer Science and Business Media LLC

Subject

Molecular Biology,Structural Biology

Link

https://www.nature.com/articles/s41594-022-00796-6.pdf

Reference52 articles.

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3. Grailhe, R. et al. Increased exploratory activity and altered response to LSD in mice lacking the 5-HT5A receptor. Neuron 22, 581–591 (1999).

4. Pierce, P. A., Xie, G. X., Levine, J. D. & Peroutka, S. J. 5-Hydroxytryptamine receptor subtype messenger RNAs in rat peripheral sensory and sympathetic ganglia: a polymerase chain reaction study. Neuroscience 70, 553–559 (1996).

5. Sagi, Y. et al. Emergence of 5-HT5A signaling in parvalbumin neurons mediates delayed antidepressant action. Mol. Psychiatry 25, 1191–1201 (2020).

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