Human substance P receptor binding mode of the antagonist drug aprepitant by NMR and crystallography
Author:
Publisher
Springer Science and Business Media LLC
Subject
General Physics and Astronomy,General Biochemistry, Genetics and Molecular Biology,General Chemistry
Link
http://www.nature.com/articles/s41467-019-08568-5.pdf
Reference42 articles.
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3. Quartara, L. & Maggi, C. A. The tachykinin NK1 receptor. Part II: distribution and pathophysiological roles. Neuropeptides 32, 1–49 (1998).
4. Iversen, L. Substance P equals pain substance? Nature 392, 334–335 (1998).
5. Kramer, M. S. et al. Distinct mechanism for antidepressant activity by blockade of central substance P receptors. Science 281, 1640–1645 (1998).
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