Human native kappa opioid receptor functions not predicted by recombinant receptors: Implications for drug design-Reference-Cited by-同舟云学术

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Human native kappa opioid receptor functions not predicted by recombinant receptors: Implications for drug design

Published:2016-08 Issue:1 Volume:6 Page:
ISSN:2045-2322
Container-title:Scientific Reports
language:en
Short-container-title:Sci Rep

Author:

Broad John,Maurel Damien,Kung Victor W. S.,Hicks Gareth A.,Schemann Michael,Barnes Michael R.,Kenakin Terrence P.,Granier Sébastien,Sanger Gareth J.

Publisher

Springer Science and Business Media LLC

Subject

Multidisciplinary

Link

http://www.nature.com/articles/srep30797.pdf

Reference70 articles.

1. Zhou, L. et al. Development of functionally selective, small molecule agonists at kappa opioid receptors. J. Biol. Chem. 288, 36703–36716 (2013).

2. Bourgeois, C. et al. Synthesis and pharmacological evaluation of 5-pyrrolidinylquinoxalines as a novel class of peripherally restricted κ-opioid receptor agonists. J. Med. Chem. 57, 6845–6860 (2014).

3. Cheng, M. F. et al. Discovery, structure-activity relationship studies, and anti-nociceptive effects of 1-phenyl-3,6,6-trimethyl-1,5,6,7-tetrahydro-4H-indazol-4-one as novel opioid receptor agonists. Bioorg. Med. Chem. 22, 4694–4703 (2014).

4. White, K. L. et al. Identification of novel functionally selective κ-opioid receptor scaffolds. Mol. Pharmacol. 85, 83–90 (2014).

5. Rivière, P. J.-M. Peripheral kappa-opioid agonists for visceral pain. Br. J. Pharmacol. 141, 1331–1334 (2004).

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