A clickable inhibitor reveals context-dependent autoactivation of p90 RSK
Author:
Publisher
Springer Science and Business Media LLC
Subject
Cell Biology,Molecular Biology
Link
http://www.nature.com/articles/nchembio859.pdf
Reference30 articles.
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3. Smith, J.A., Poteet-Smith, C.E., Malarkey, K. & Sturgill, T.W. Identification of an extracellular signal-regulated kinase (ERK) docking site in ribosomal S6 kinase, a sequence critical for activation by ERK in vivo. J. Biol. Chem. 274, 2893–2898 (1999).
4. Gavin, A.C. & Nebreda, A.R.A. MAP kinase docking site is required for phosphorylation and activation of p90(rsk)/MAPKAP kinase-1. Curr. Biol. 9, 281–284 (1999).
5. Frodin, M., Jensen, C.J., Merienne, K. & Gammeltoft, S. A phosphoserine-regulated docking site in the protein kinase RSK2 that recruits and activates PDK1. EMBO J. 19, 2924–2934 (2000).
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