A chemical probe selectively inhibits G9a and GLP methyltransferase activity in cells-Reference-Cited by-同舟云学术

A chemical probe selectively inhibits G9a and GLP methyltransferase activity in cells

Published:2011-07-10 Issue:8 Volume:7 Page:566-574
ISSN:1552-4450
Container-title:Nature Chemical Biology
language:en
Short-container-title:Nat Chem Biol

Author:

Vedadi Masoud,Barsyte-Lovejoy Dalia,Liu Feng,Rival-Gervier Sylvie,Allali-Hassani Abdellah,Labrie Viviane,Wigle Tim J,DiMaggio Peter A,Wasney Gregory A,Siarheyeva Alena,Dong Aiping,Tempel Wolfram,Wang Sun-Chong,Chen Xin,Chau Irene,Mangano Thomas J,Huang Xi-ping,Simpson Catherine D,Pattenden Samantha G,Norris Jacqueline L,Kireev Dmitri B,Tripathy Ashutosh,Edwards Aled,Roth Bryan L,Janzen William P,Garcia Benjamin A,Petronis Arturas,Ellis James,Brown Peter J,Frye Stephen V,Arrowsmith Cheryl H,Jin Jian

Publisher

Springer Science and Business Media LLC

Subject

Cell Biology,Molecular Biology

Link

http://www.nature.com/articles/nchembio.599.pdf

Reference50 articles.

1. Kouzarides, T. Chromatin modifications and their function. Cell 128, 693–705 (2007).

2. Martin, C. & Zhang, Y. The diverse functions of histone lysine methylation. Nat. Rev. Mol. Cell Biol. 6, 838–849 (2005).

3. Jenuwein, T. & Allis, C.D. Translating the histone code. Science 293, 1074–1080 (2001).

4. Bernstein, B.E., Meissner, A. & Lander, E.S. The mammalian epigenome. Cell 128, 669–681 (2007).

5. Gelato, K.A. & Fischle, W. Role of histone modifications in defining chromatin structure and function. Biol. Chem. 389, 353–363 (2008).

Cited by 459 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. A Live‐Cell Epigenome Manipulation by Photo‐Stimuli‐Responsive Histone Methyltransferase Inhibitor;Advanced Science;2024-09-09

2. Structure-based development of novel substrate-type G9a inhibitors as epigenetic modulators for sickle cell disease treatment;Bioorganic & Medicinal Chemistry Letters;2024-09

3. A First-in-Class High-Throughput Screen to Discover Modulators of the Alternative Lengthening of Telomeres (ALT) Pathway;ACS Pharmacology & Translational Science;2024-08-13

4. Newly developed oral bioavailable EHMT2 inhibitor as a potential epigenetic therapy for Prader-Willi syndrome;Molecular Therapy;2024-08

5. Discovery of Potent and Selective G9a Degraders for the Treatment of Pancreatic Cancer;Journal of Medicinal Chemistry;2024-07-23