Binding kinetics of cariprazine and aripiprazole at the dopamine D3 receptor
Author:
Publisher
Springer Science and Business Media LLC
Subject
Multidisciplinary
Link
http://www.nature.com/articles/s41598-018-30794-y.pdf
Reference40 articles.
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3. Ágai-Csongor, É. et al. Discovery of cariprazine (RGH-188): a novel antipsychotic acting on dopamine D3/D2 receptors. Bioorg. Med. Chem. Lett. 22, 3437–3440 (2012).
4. Wesołowska, A., Partyka, A., Jastrzębska-Więsek, M. & Kołaczkowski, M. The preclinical discovery and development of cariprazine for the treatment of schizophrenia. Expert Opin. Drug Discov. in press, 1471057; https://doi.org/10.1080/17460441.2018.1471057 (2018).
5. Németh, G. et al. Cariprazine versus risperidone monotherapy for treatment of predominant negative symptoms in patients with schizophrenia: a randomised, double-blind, controlled trial. Lancet 389, 1103–1113 (2017).
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