High-throughput screening of the Plasmodium falciparum cGMP-dependent protein kinase identified a thiazole scaffold which kills erythrocytic and sexual stage parasites-Reference-Cited by-同舟云学术

High-throughput screening of the Plasmodium falciparum cGMP-dependent protein kinase identified a thiazole scaffold which kills erythrocytic and sexual stage parasites

Published:2019-05-07 Issue:1 Volume:9 Page:
ISSN:2045-2322
Container-title:Scientific Reports
language:en
Short-container-title:Sci Rep

Author:

Penzo Maria,de las Heras-Dueña Laura,Mata-Cantero Lydia,Diaz-Hernandez Beatriz,Vazquez-Muñiz Maria-Jesus,Ghidelli-Disse Sonja,Drewes Gerard,Fernandez-Alvaro Elena,Baker David A.^ORCID

Publisher

Springer Science and Business Media LLC

Subject

Multidisciplinary

Link

http://www.nature.com/articles/s41598-019-42801-x.pdf

Reference61 articles.

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3. Dondorp, A. M. et al. Artemisinin resistance in Plasmodium falciparum malaria. N Engl J Med 361, 455–467, https://doi.org/10.1056/NEJMoa0808859 (2009).

4. Noedl, H., Socheat, D. & Satimai, W. Artemisinin-resistant malaria in Asia. N Engl J Med 361, 540–541, https://doi.org/10.1056/NEJMc0900231 (2009).

5. Mukherjee, A. et al. Artemisinin resistance without pfkelch13 mutations in Plasmodium falciparum isolates from Cambodia. Malar J 16, 195, https://doi.org/10.1186/s12936-017-1845-5 (2017).

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