Novel selective, potent naphthyl TRPM8 antagonists identified through a combined ligand- and structure-based virtual screening approach-Reference-Cited by-同舟云学术

Novel selective, potent naphthyl TRPM8 antagonists identified through a combined ligand- and structure-based virtual screening approach

Published:2017-09-08 Issue:1 Volume:7 Page:
ISSN:2045-2322
Container-title:Scientific Reports
language:en
Short-container-title:Sci Rep

Author:

Beccari Andrea R.,Gemei Marica,Lo Monte Matteo,Menegatti Nazareno,Fanton Marco,Pedretti Alessandro,Bovolenta Silvia,Nucci Cinzia,Molteni Angela,Rossignoli Andrea,Brandolini Laura,Taddei Alessandro,Za Lorena,Liberati Chiara,Vistoli Giulio

Publisher

Springer Science and Business Media LLC

Subject

Multidisciplinary

Link

http://www.nature.com/articles/s41598-017-11194-0.pdf

Reference80 articles.

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3. Ramsey, I. S., Delling, M. & Clapham, D. E. An introduction to TRP channels. Annu Rev Physiol 68, 619–647, doi:10.1146/annurev.physiol.68.040204.100431 (2006).

4. Vay, L., Gu, C. & McNaughton, P. A. The thermo-TRP ion channel family: properties and therapeutic implications. Br J Pharmacol 165, 787–801, doi:10.1111/j.1476-5381.2011.01601.x (2012).

5. Nilius, B. & Owsianik, G. The transient receptor potential family of ion channels. Genome Biol 12, 218, doi:10.1186/gb-2011-12-3-218 (2011).

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