Rational drug-design approach supported with thermodynamic studies — a peptide leader for the efficient bi-substrate inhibitor of protein kinase CK2
Author:
Funder
Narodowe Centrum Nauki
Publisher
Springer Science and Business Media LLC
Subject
Multidisciplinary
Link
http://www.nature.com/articles/s41598-019-47404-0.pdf
Reference47 articles.
1. Hanks, S. K. & Hunter, T. Protein kinases 6. The eukaryotic protein kinase superfamily: kinase (catalytic) domain structure and classification. Faseb j 9, 576–596 (1995).
2. Fabbro, D. et al. Protein kinases as targets for anticancer agents: from inhibitors to useful drugs. Pharmacology & Therapeutics 93, 79–98, https://doi.org/10.1016/S0163-7258(02)00179-1 (2002).
3. Fabbro, D. & Garcia-Echeverria, C. Targeting protein kinases in cancer therapy. Current Opinion in Drug Discovery & Development 5, 701–712 (2002).
4. Bhullar, K. S. et al. Kinase-targeted cancer therapies: progress, challenges and future directions. Molecular cancer 17, 48–48 (2018).
5. Kennelly, P. J. & Krebs, E. G. Consensus sequences as substrate specificity determinants for protein kinases and protein phosphatases. Journal of Biological Chemistry 266, 15555–15558 (1991).
Cited by 10 articles. 订阅此论文施引文献 订阅此论文施引文献,注册后可以免费订阅5篇论文的施引文献,订阅后可以查看论文全部施引文献
1. Structure‐Guided Drug Design Targeting Abl Kinase: How Structure and Regulation Can Assist in Designing New Drugs;ChemBioChem;2024-09-12
2. Designing drugs and chemical probes with the dualsteric approach;Chemical Society Reviews;2023
3. Microscale thermophoresis as a powerful growing analytical technique for the investigation of biomolecular interaction and the determination of binding parameters;Methods and Applications in Fluorescence;2022-07-28
4. 5,6-diiodo-1H-benzotriazole: new TBBt analogue that minutely affects mitochondrial activity;Scientific Reports;2021-12
5. Correlation Analysis of Target Selectivity and Side Effects of FDA‐Approved Kinase Inhibitors**;ChemistrySelect;2021-08-13
1.学者识别学者识别
2.学术分析学术分析
3.人才评估人才评估
"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370
www.globalauthorid.com
TOP
Copyright © 2019-2024 北京同舟云网络信息技术有限公司 京公网安备11010802033243号 京ICP备18003416号-3