Ligands of the antiestrogen-binding site induce active cell death and autophagy in human breast cancer cells through the modulation of cholesterol metabolism-Reference-Cited by-同舟云学术

Ligands of the antiestrogen-binding site induce active cell death and autophagy in human breast cancer cells through the modulation of cholesterol metabolism

Published:2009-06-12 Issue:10 Volume:16 Page:1372-1384
ISSN:1350-9047
Container-title:Cell Death & Differentiation
language:en
Short-container-title:Cell Death Differ

Author:

de Medina P,Payré B,Boubekeur N,Bertrand-Michel J,Tercé F,Silvente-Poirot S,Poirot M

Publisher

Springer Science and Business Media LLC

Subject

Cell Biology,Molecular Biology

Link

http://www.nature.com/articles/cdd200962.pdf

Reference37 articles.

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2. Kedjouar B, De Medina P, Oulad-Abdelghani M, Payre B, Silvente-Poirot S, Favre G et al. Molecular characterization of the microsomal tamoxifen binding site. J Biol Chem 2004; 279: 34048–34061.

3. Brandes LJ . A diphenylmethane derivative selective for the anti-estrogen binding site may help define its biological role. Biochem Biophys Res Commun 1984; 124: 244–249.

4. Poirot M, De Medina P, Delarue F, Perie JJ, Klaebe A, Faye JC . Synthesis, binding and structure–affinity studies of new ligands for the microsomal anti-estrogen binding site (AEBS). Bioorg Med Chem 2000; 8: 2007–2016.

5. de Medina P, Favre G, Poirot M . Multiple targeting by the antitumor drug tamoxifen: a structure–activity study. Curr Med Chem Anticancer Agents 2004; 4: 491–508.

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