Adding calorimetric data to decision making in lead discovery: a hot tip
Author:
Publisher
Springer Science and Business Media LLC
Subject
Drug Discovery,Pharmacology,General Medicine
Link
http://www.nature.com/articles/nrd3054.pdf
Reference31 articles.
1. Ladbury, J. E. Counting the calories to stay in the groove. Structure 3, 635–639 (1995).
2. Ladbury, J. E. & Chowdhry, B. Z. Sensing the heat: the application of isothermal titration calorimetry to thermodynamic studies of biomolecular interactions. Chem. Biol. 3, 791–801 (1996).
3. Ladbury, J. E. Isothermal titration calorimetry: application to structure-based drug design. Thermochim. Acta 380, 209–215 (2001).
4. Velazquez-Campoy, A. & Freire, E. ITC in the post-genomic era...? Priceless. Biophys. Chem. 115, 115–124 (2005).
5. Freire, E. in Proteomics and Protein–Protein Interactions: Biology, Chemistry, Bioinformatics, and Drug Design. Vol. 3 (ed. Waksman, G.) 291–307 (Springer, New York, 2005).
Cited by 343 articles. 订阅此论文施引文献 订阅此论文施引文献,注册后可以免费订阅5篇论文的施引文献,订阅后可以查看论文全部施引文献
1. Functional study of a lytic polysaccharide monooxygenase MsLPMO3 from Morchella sextelata in the oxidative degradation of cellulose;Enzyme and Microbial Technology;2024-02
2. Accurate calculation of affinity changes to the close state of influenza A M2 transmembrane domain in response to subtle structural changes of adamantyl amines using free energy perturbation methods in different lipid bilayers;Biochimica et Biophysica Acta (BBA) - Biomembranes;2024-02
3. An isothermal calorimetry assay for determining steady state kinetic and enzyme inhibition parameters for SARS-CoV-2 3CL-protease;2024-01-31
4. A miniaturized mode-of-action profiling platform enables high throughput characterization of the molecular and cellular dynamics of EZH2 inhibition;Scientific Reports;2024-01-19
5. Alcohol‐Induced Conformation Changes and Thermodynamic Signatures in the Binding of Polyphenols to Proline‐Rich Salivary Proteins;Chemistry – A European Journal;2023-10-24
1.学者识别学者识别
2.学术分析学术分析
3.人才评估人才评估
"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370
www.globalauthorid.com
TOP
Copyright © 2019-2024 北京同舟云网络信息技术有限公司 京公网安备11010802033243号 京ICP备18003416号-3