A tetraoxane-based antimalarial drug candidate that overcomes PfK13-C580Y dependent artemisinin resistance
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Published:2017-05-24
Issue:1
Volume:8
Page:
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ISSN:2041-1723
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Container-title:Nature Communications
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language:en
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Short-container-title:Nat Commun
Author:
O’Neill Paul M., Amewu Richard K., Charman Susan A., Sabbani Sunil, Gnädig Nina F., Straimer Judith, Fidock David A.ORCID, Shore Emma R., Roberts Natalie L., Wong Michael H.-L., Hong W. David, Pidathala Chandrakala, Riley Chris, Murphy Ben, Aljayyoussi Ghaith, Gamo Francisco Javier, Sanz Laura, Rodrigues Janneth, Cortes Carolina Gonzalez, Herreros Esperanza, Angulo-Barturén Iñigo, Jiménez-Díaz María Belén, Bazaga Santiago Ferrer, Martínez-Martínez María Santos, Campo Brice, Sharma Raman, Ryan Eileen, Shackleford David M., Campbell Simon, Smith Dennis A., Wirjanata Grennady, Noviyanti Rintis, Price Ric N., Marfurt Jutta, Palmer Michael J., Copple Ian M., Mercer Amy E., Ruecker Andrea, Delves Michael J., Sinden Robert E., Siegl Peter, Davies Jill, Rochford Rosemary, Kocken Clemens H. M., Zeeman Anne-Marie, Nixon Gemma L., Biagini Giancarlo A., Ward Stephen A.
Publisher
Springer Science and Business Media LLC
Subject
General Physics and Astronomy,General Biochemistry, Genetics and Molecular Biology,General Chemistry
Reference46 articles.
1. WHO. Global Report on Antimalarial Drug Efficacy and Drug Resistance: 2000–2010 (WHO, 2010). 2. WHO. Guidelines for the Treatment of Malaria 2nd edn (WHO, 2010). 3. Wells, T. N., van Huijsduijnen, R. H. & Van Voorhis, W. C. Malaria medicines: a glass half full? Nat. Rev. Drug. Discov. 14, 424–442 (2015). 4. Noedl, H. et al. Evidence of artemisinin-resistant malaria in western Cambodia. N. Engl. J. Med. 359, 2619–2620 (2008). 5. Dondorp, A. M. et al. Artemisinin resistance in Plasmodium falciparum malaria. N. Engl. J. Med. 361, 455–467 (2009).
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