Analysis of the pharmacokinetic/pharmacodynamic relationship of a small molecule CXCR3 antagonist, NBI-74330, using a murine CXCR3 internalization assay
Author:
Publisher
Wiley
Subject
Pharmacology
Link
http://onlinelibrary.wiley.com/wol1/doi/10.1038/sj.bjp.0707519/fullpdf
Reference51 articles.
1. Dissociation of chemotaxis from agonist-induced receptor internalization in a lymphocyte cell line transfected with CCR2B. Evidence that directed migration does not require rapid modulation of signaling at the receptor level;Arai;J Biol Chem,1997
2. Functional evidence equating the pharmacologically-defined alpha 1A- and cloned alpha 1C-adrenoceptor: studies in the isolated perfused kidney of rat;Blue;Br J Pharmacol,1995
3. Differential expression of chemokine receptors and chemotactic responsiveness of type 1 T helper cells (Th1s) and Th2s;Bonecchi;J Exp Med,1998
4. CXCR3 and heparin binding sites of the chemokine IP-10 (CXCL10);Campanella;J Biol Chem,2003
5. The use of kinetic-dynamic interactions in the evaluation of drugs;Campbell;Psychopharmacology (Berl),1990
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