XP13512 [(±)-1-([(α-Isobutanoyloxyethoxy)carbonyl] aminomethyl)-1-cyclohexane Acetic Acid], A Novel Gabapentin Prodrug: I. Design, Synthesis, Enzymatic Conversion to Gabapentin, and Transport by Intestinal Solute Transporters-Reference-Cited by-同舟云学术

XP13512 [(±)-1-([(α-Isobutanoyloxyethoxy)carbonyl] aminomethyl)-1-cyclohexane Acetic Acid], A Novel Gabapentin Prodrug: I. Design, Synthesis, Enzymatic Conversion to Gabapentin, and Transport by Intestinal Solute Transporters

Published:2004-05-14 Issue:1 Volume:311 Page:315-323
ISSN:0022-3565
Container-title:Journal of Pharmacology and Experimental Therapeutics
language:en
Short-container-title:J Pharmacol Exp Ther

Author:

Cundy Kenneth C.,Branch Russell,Chernov-Rogan Tania,Dias Tracy,Estrada Toño,Hold Karin,Koller Kerry,Liu Xiaoli,Mann Adam,Panuwat Matt,Raillard Stephen P.,Upadhyay Shubhra,Wu Quincey Q.,Xiang Jia-Ning,Yan Hui,Zerangue Noa,Zhou Cindy X.,Barrett Ronald W.,Gallop Mark A.

Publisher

American Society for Pharmacology & Experimental Therapeutics (ASPET)

Subject

Pharmacology,Molecular Medicine

Reference41 articles.

1. (Acyloxy)alkyl carbamates as novel bioreversible prodrugs for amines: increased permeation through biological membranes

2. Gabapentin for the Symptomatic Treatment of Painful Neuropathy in Patients With Diabetes MellitusA Randomized Controlled Trial

3. Biotin absorption from the hindgut of the pig

4. The absorption of gabapentin following high dose escalation

5. Effects of Age and Gender on Single-Dose Pharmacokinetics of Gabapentin

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