Phenylalanine-544 Plays a Key Role in Substrate and Inhibitor Binding by Providing a Hydrophobic Packing Point at the Active Site of Insulin-Regulated Aminopeptidase-Reference-Cited by-同舟云学术

Phenylalanine-544 Plays a Key Role in Substrate and Inhibitor Binding by Providing a Hydrophobic Packing Point at the Active Site of Insulin-Regulated Aminopeptidase

Published:2010-07-13 Issue:4 Volume:78 Page:600-607
ISSN:0026-895X
Container-title:Molecular Pharmacology
language:en
Short-container-title:Mol Pharmacol

Author:

Albiston Anthony L.,Pham Vi,Ye Siying,Ng Leelee,Lew Rebecca A.,Thompson Philip E.,Holien Jessica K.,Morton Craig J.,Parker Michael W.,Chai Siew Yeen

Publisher

American Society for Pharmacology & Experimental Therapeutics (ASPET)

Subject

Pharmacology,Molecular Medicine

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5. Ligands to the (IRAP)/AT4 receptor encompassing a 4-hydroxydiphenylmethane scaffold replacing Tyr2

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