Michaelis-Menten quantification of ligand signalling bias applied to the promiscuous Vasopressin V2 receptor
Author:
Publisher
American Society for Pharmacology & Experimental Therapeutics (ASPET)
Subject
Pharmacology,Molecular Medicine
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1. Functional consequences of spatial, temporal and ligand bias of G protein-coupled receptors;Nature Reviews Nephrology;2024-07-22
2. G protein–coupled receptor endocytosis generates spatiotemporal bias in β-arrestin signaling;Science Signaling;2024-06-25
3. β-Arrestin-dependent and -independent endosomal G protein activation by the vasopressin type 2 receptor;eLife;2023-10-19
4. β-Arrestin-dependent and -independent endosomal G protein activation by the vasopressin type 2 receptor;eLife;2023-10-19
5. Allosteric modulation of G protein-coupled receptors as a novel therapeutic strategy in neuropathic pain;Acta Pharmaceutica Sinica B;2023-07
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