Degraders: The Ultimate Weapon Against Amplified Driver Kinases in Cancer
Author:
Publisher
American Society for Pharmacology & Experimental Therapeutics (ASPET)
Subject
Pharmacology,Molecular Medicine
Reference96 articles.
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2. Mutant-selective degradation by BRAF-targeting PROTACs;Alabi;Nat Commun,2021
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1. Selective Degradation of MLK3 by a Novel CEP1347-VHL-02 PROTAC Compound Limits the Oncogenic Potential of TNBC;Journal of Medicinal Chemistry;2024-08-29
2. PIM1 targeted degradation prevents the emergence of chemoresistance in prostate cancer;Cell Chemical Biology;2023-11
3. Bifunctional degraders of cyclin dependent kinase 9 (CDK9): Probing the relationship between linker length, properties, and selective protein degradation;European Journal of Medicinal Chemistry;2023-06
4. Measurement and utilization of the proteomic reactivity by mass spectrometry;Mass Spectrometry Reviews;2023-03-16
5. Kinase-targeting small-molecule inhibitors and emerging bifunctional molecules;Trends in Pharmacological Sciences;2022-10
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