Preclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive Disorder-Reference-Cited by-同舟云学术

Preclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive Disorder

Published:2017-09-27 Issue:3 Volume:363 Page:377-393
ISSN:0022-3565
Container-title:Journal of Pharmacology and Experimental Therapeutics
language:en
Short-container-title:J Pharmacol Exp Ther

Author:

Bristow Linda J.,Gulia Jyoti,Weed Michael R.,Srikumar Bettadapura N.,Li Yu-Wen,Graef John D.,Naidu Pattipati S.,Sanmathi Charulatha,Aher Jayant,Bastia Tanmaya,Paschapur Mahesh,Kalidindi Narasimharaju,Kumar Kuchibhotla Vijaya,Molski Thaddeus,Pieschl Rick,Fernandes Alda,Brown Jeffrey M.,Sivarao Digavalli V.,Newberry Kimberly,Bookbinder Mark,Polino Joseph,Keavy Deborah,Newton Amy,Shields Eric,Simmermacher Jean,Kempson James,Li Jianqing,Zhang Huiping,Mathur Arvind,Kallem Raja Reddy,Sinha Meenakshee,Ramarao Manjunath,Vikramadithyan Reeba K.,Thangathirupathy Srinivasan,Warrier Jayakumar,Islam Imadul,Bronson Joanne J.,Olson Richard E.,Macor John E.,Albright Charlie F.,King Dalton,Thompson Lorin A.,Marcin Lawrence R.,Sinz Michael

Publisher

American Society for Pharmacology & Experimental Therapeutics (ASPET)

Subject

Pharmacology,Molecular Medicine

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