Impact of Impurity on Kinetic Estimates from Transport and Inhibition Studies
Author:
Publisher
American Society for Pharmacology & Experimental Therapeutics (ASPET)
Subject
Pharmacology,Molecular Medicine
Reference12 articles.
1. Bias in Estimation of Transporter Kinetic Parameters from Overexpression Systems: Interplay of Transporter Expression Level and Substrate Affinity
2. Apical Sodium Dependent Bile Acid Transporter (ASBT, SLC10A2): A Potential Prodrug Target
3. Development of Stably Transfected Monolayer Overexpressing the Human Apical Sodium-Dependent Bile Acid Transporter (hASBT)
4. Influence of Charge and Steric Bulk in the C-24 Region on the Interaction of Bile Acids with Human Apical Sodium-Dependent Bile Acid Transporter
5. Interaction of Native Bile Acids with Human Apical Sodium-Dependent Bile Acid Transporter (hASBT): Influence of Steroidal Hydroxylation Pattern and C-24 Conjugation
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1. Structural Requirements of the Human Sodium-Dependent Bile Acid Transporter (hASBT): Role of 3- and 7-OH Moieties on Binding and Translocation of Bile Acids;Molecular Pharmaceutics;2013-12-26
2. Structural requirements of bile acid transporters: C-3 and C-7 modifications of steroidal hydroxyl groups;European Journal of Pharmaceutical Sciences;2012-05
3. Synthesis and Pharmacological Evaluation of 4-Iminothiazolidinones for Inhibition of PI3 Kinase;Australian Journal of Chemistry;2012
4. Structural Requirements of the ASBT by 3D-QSAR Analysis Using Aminopyridine Conjugates of Chenodeoxycholic Acid;Bioconjugate Chemistry;2010-10-22
5. Synthesis and in vitro evaluation of potential sustained release prodrugs via targeting ASBT;International Journal of Pharmaceutics;2010-08-30
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