Identification and Characterization of INCB9471, an Allosteric Noncompetitive Small-Molecule Antagonist of C-C Chemokine Receptor 5 with Potent Inhibitory Activity against Monocyte Migration and HIV-1 Infection-Reference-Cited by-同舟云学术

Identification and Characterization of INCB9471, an Allosteric Noncompetitive Small-Molecule Antagonist of C-C Chemokine Receptor 5 with Potent Inhibitory Activity against Monocyte Migration and HIV-1 Infection

Published:2011-04-01 Issue:1 Volume:338 Page:228-239
ISSN:0022-3565
Container-title:Journal of Pharmacology and Experimental Therapeutics
language:en
Short-container-title:J Pharmacol Exp Ther

Author:

Shin Niu,Solomon Kim,Zhou Naiming,Wang Kathy He,Garlapati Vasudha,Thomas Beth,Li Yanlong,Covington Maryanne,Baribaud Frederic,Erickson-Viitanen Susan,Czerniak Phil,Contel Nancy,Liu Phillip,Burn Timothy,Hollis Gregory,Yeleswaram Swamy,Vaddi Kris,Xue Chu-Biao,Metcalf Brian,Friedman Steve,Scherle Peggy,Newton Robert

Publisher

American Society for Pharmacology & Experimental Therapeutics (ASPET)

Subject

Pharmacology,Molecular Medicine

Reference41 articles.

1. The Role of CC Chemokine Receptor 5 (CCR5) in Islet Allograft Rejection

2. Characterization of chemokines and their receptors in the central nervous system: physiopathological implications

3. Baroudy BM Clasder JW Josien HB McCombie SW McKittrick BA Miller MW Neustadt BR Palani A Smith EM Steensma R . (2000), inventors

4. Schering-Plough Corp., assignee. Piperazine derivatives useful as CCR5 antagonists. World patent WO200006558. 2000 Sep 11.

5. CCR5 deficiency decreases susceptibility to experimental cerebral malaria

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