Development of a Highly Selective Allosteric Antagonist Radioligand for the Type 1 Cholecystokinin Receptor and Elucidation of Its Molecular Basis of Binding-Reference-Cited by-同舟云学术

Development of a Highly Selective Allosteric Antagonist Radioligand for the Type 1 Cholecystokinin Receptor and Elucidation of Its Molecular Basis of Binding

Published:2014-10-15 Issue:1 Volume:87 Page:130-140
ISSN:0026-895X
Container-title:Molecular Pharmacology
language:en
Short-container-title:Mol Pharmacol

Author:

Dong Maoqing^ORCID,Vattelana Ashton M.,Lam Polo C.-H.,Orry Andrew J.,Abagyan Ruben,Christopoulos Arthur,Sexton Patrick M.^ORCID,Haines David R.,Miller Laurence J.

Publisher

American Society for Pharmacology & Experimental Therapeutics (ASPET)

Subject

Pharmacology,Molecular Medicine

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1. Biased Probability Monte Carlo Conformational Searches and Electrostatic Calculations for Peptides and Proteins

2. ICM?A new method for protein modeling and design: Applications to docking and structure prediction from the distorted native conformation

3. Helix movement is coupled to displacement of the second extracellular loop in rhodopsin activation

4. Synthesis and in Vitro Characterization of Radioiodinatable Benzodiazepines Selective for Type 1 and Type 2 Cholecystokinin Receptors

5. Key Differences in Molecular Complexes of the Cholecystokinin Receptor with Structurally Related Peptide Agonist, Partial Agonist, and Antagonist

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