In Vivo Characterization of the Ultrapotent Monoacylglycerol Lipase Inhibitor (1H-1,2,4-triazol-1-yl)methanone (JJKK-048)-Reference-Cited by-同舟云学术

In Vivo Characterization of the Ultrapotent Monoacylglycerol Lipase Inhibitor (1H-1,2,4-triazol-1-yl)methanone (JJKK-048)

Published:2016-07-22 Issue:1 Volume:359 Page:62-72
ISSN:1521-0103
Container-title:Journal of Pharmacology and Experimental Therapeutics
language:en
Short-container-title:Journal of Pharmacology and Experimental Therapeutics

Author:

Aaltonen N.,Kedzierska E.,Orzelska-Gorka J.,Lehtonen M.,Navia-Paldanius D.,Jakupovic H.,Savinainen J. R.,Nevalainen T.,Laitinen J. T.,Parkkari T.,Gynther M.

Publisher

American Society for Pharmacology & Experimental Therapeutics (ASPET)

Subject

Pharmacology,Molecular Medicine

Reference52 articles.

1. Brain regional cannabinoid CB1 receptor signalling and alternative enzymatic pathways for 2-arachidonoylglycerol generation in brain sections of diacylglycerol lipase deficient mice

2. Piperazine and Piperidine Triazole Ureas as Ultrapotent and Highly Selective Inhibitors of Monoacylglycerol Lipase

3. Novel Mechanistic Class of Fatty Acid Amide Hydrolase Inhibitors with Remarkable Selectivity

4. Mechanism of Carbamate Inactivation of FAAH: Implications for the Design of Covalent Inhibitors and In Vivo Functional Probes for Enzymes

5. Actions of the dual FAAH/MAGL inhibitor JZL195 in a murine inflammatory pain model

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