A New Molecular Mechanism To Engineer Protean Agonism at a G Protein–Coupled Receptor-Reference-Cited by-同舟云学术

A New Molecular Mechanism To Engineer Protean Agonism at a G Protein–Coupled Receptor

Published:2017-02-06 Issue:4 Volume:91 Page:348-356
ISSN:0026-895X
Container-title:Molecular Pharmacology
language:en
Short-container-title:Mol Pharmacol

Author:

De Min Anna,Matera Carlo,Bock Andreas,Holze Janine,Kloeckner Jessica,Muth Mathias,Traenkle Christian,De Amici Marco,Kenakin Terry,Holzgrabe Ulrike,Dallanoce Clelia,Kostenis Evi,Mohr Klaus,Schrage Ramona

Publisher

American Society for Pharmacology & Experimental Therapeutics (ASPET)

Subject

Pharmacology,Molecular Medicine

Reference65 articles.

1. Dualsteric GPCR targeting: a novel route to binding and signaling pathway selectivity

2. Influence of sodium substitutes on 5-HT-mediated effects at mouse 5-HT3receptors

3. Hill coefficients and the logistic equation

4. Modulation of Gq-Protein-Coupled Inositol Trisphosphate and Ca2+ Signaling by the Membrane Potential

5. Ligand Binding Ensembles Determine Graded Agonist Efficacies at a G Protein-coupled Receptor

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