Extracellular Loop 2 of the Adenosine A1 Receptor Has a Key Role in Orthosteric Ligand Affinity and Agonist Efficacy-Reference-Cited by-同舟云学术

Extracellular Loop 2 of the Adenosine A1 Receptor Has a Key Role in Orthosteric Ligand Affinity and Agonist Efficacy

Published:2016-09-28 Issue:6 Volume:90 Page:703-714
ISSN:0026-895X
Container-title:Molecular Pharmacology
language:en
Short-container-title:Mol Pharmacol

Author:

Nguyen Anh T.N.,Baltos Jo-Anne,Thomas Trayder,Nguyen Toan D.,Muñoz Laura López,Gregory Karen J.,White Paul J.,Sexton Patrick M.,Christopoulos Arthur,May Lauren T.

Publisher

American Society for Pharmacology & Experimental Therapeutics (ASPET)

Subject

Pharmacology,Molecular Medicine

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4. [19] Integrated methods for the construction of three-dimensional models and computational probing of structure-function relations in G protein-coupled receptors

5. Quantification of adenosine A 1 receptor biased agonism: Implications for drug discovery

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