N-((1S)-1-{[4-((2S)-2-{[(2,4-Dichlorophenyl)sulfonyl]amino}-3-hydroxypropanoyl)-1-piperazinyl]carbonyl}-3-methylbutyl)-1-benzothiophene-2-carboxamide (GSK1016790A), a Novel and Potent Transient Receptor Potential Vanilloid 4 Channel Agonist Induces Urinary Bladder Contraction and Hyperactivity: Part I-Reference-Cited by-同舟云学术

N-((1S)-1-{[4-((2S)-2-{[(2,4-Dichlorophenyl)sulfonyl]amino}-3-hydroxypropanoyl)-1-piperazinyl]carbonyl}-3-methylbutyl)-1-benzothiophene-2-carboxamide (GSK1016790A), a Novel and Potent Transient Receptor Potential Vanilloid 4 Channel Agonist Induces Urinary Bladder Contraction and Hyperactivity: Part I

Published:2008-05-22 Issue:2 Volume:326 Page:432-442
ISSN:0022-3565
Container-title:Journal of Pharmacology and Experimental Therapeutics
language:en
Short-container-title:J Pharmacol Exp Ther

Author:

Thorneloe Kevin S.,Sulpizio Anthony C.,Lin Zuojun,Figueroa David J.,Clouse Angela K.,McCafferty Gerald P.,Chendrimada Tim P.,Lashinger Erin S. R.,Gordon Earl,Evans Louise,Misajet Blake A.,DeMarini Douglas J.,Nation Josephine H.,Casillas Linda N.,Marquis Robert W.,Votta Bartholomew J.,Sheardown Steven A.,Xu Xiaoping,Brooks David P.,Laping Nicholas J.,Westfall Timothy D.

Publisher

American Society for Pharmacology & Experimental Therapeutics (ASPET)

Subject

Pharmacology,Molecular Medicine

Reference40 articles.

1. A Transient Receptor Potential Vanilloid 4-Dependent Mechanism of Hyperalgesia Is Engaged by Concerted Action of Inflammatory Mediators

2. Transient Receptor Potential Vanilloid 4–Mediated Disruption of the Alveolar Septal Barrier

3. Swelling-activated Ca2+ Entry via TRPV4 Channel Is Defective in Cystic Fibrosis Airway Epithelia

4. TRPV1 (vanilloid receptor) in the urinary tract: expression, function and clinical applications

5. Vanilloid receptor expression suggests a sensory role for urinary bladder epithelial cells

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