Implementation of a Fluorescence-Based Screening Assay Identifies Histamine H3 Receptor Antagonists Clobenpropit and Iodophenpropit as Subunit-Selective N-Methyl-d-Aspartate Receptor Antagonists-Reference-Cited by-同舟云学术

Implementation of a Fluorescence-Based Screening Assay Identifies Histamine H3 Receptor Antagonists Clobenpropit and Iodophenpropit as Subunit-Selective N-Methyl-d-Aspartate Receptor Antagonists

Published:2010-03-02 Issue:3 Volume:333 Page:650-662
ISSN:0022-3565
Container-title:Journal of Pharmacology and Experimental Therapeutics
language:en
Short-container-title:J Pharmacol Exp Ther

Author:

Hansen Kasper B.,Mullasseril Praseeda,Dawit Sara,Kurtkaya Natalie L.,Yuan Hongjie,Vance Katie M.,Orr Anna G.,Kvist Trine,Ogden Kevin K.,Le Phuong,Vellano Kimberly M.,Lewis Iestyn,Kurtkaya Serdar,Du Yuhong,Qui Min,Murphy T. J.,Snyder James P.,Bräuner-Osborne Hans,Traynelis Stephen F.

Publisher

American Society for Pharmacology & Experimental Therapeutics (ASPET)

Subject

Pharmacology,Molecular Medicine

Reference40 articles.

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2. Enhancement by histamine of NMDA-mediated synaptic transmission in the hippocampus

3. Ligands for Glutamate Receptors: Design and Therapeutic Prospects

4. Histamine Potentiates N-Methyl-d-aspartate Receptors by Interacting with an Allosteric Site Distinct from the Polyamine Binding Site

5. Optimal expression of cloned NMDAR1/NMDAR2A heteromeric glutamate receptors: a biochemical characterization

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