The Biotransformation of Prasugrel, a New Thienopyridine Prodrug, by the Human Carboxylesterases 1 and 2-Reference-Cited by-同舟云学术

The Biotransformation of Prasugrel, a New Thienopyridine Prodrug, by the Human Carboxylesterases 1 and 2

Published:2008-03-27 Issue:7 Volume:36 Page:1227-1232
ISSN:0090-9556
Container-title:Drug Metabolism and Disposition
language:en
Short-container-title:Drug Metab Dispos

Author:

Williams Eric T.,Jones Karen O.,Ponsler G. Douglas,Lowery Shane M.,Perkins Everett J.,Wrighton Steven A.,Ruterbories Kenneth J.,Kazui Miho,Farid Nagy A.

Publisher

American Society for Pharmacology & Experimental Therapeutics (ASPET)

Subject

Pharmaceutical Science,Pharmacology

Reference28 articles.

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2. Structural basis of heroin and cocaine metabolism by a promiscuous human drug-processing enzyme

3. A comparison of prasugrel and clopidogrel loading doses on platelet function: magnitude of platelet inhibition is related to active metabolite formation

4. Copeland RA (1996) Enzymes: A Practical Introduction to Structure, Mechanism, and Data Analysis, Wiley-VCH, New York.

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